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Found 2 Enz. Inhib. hit(s) for PDB: 2ETM
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182010(7-(pyridin-2-yl)-N-(2,4,6-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against FAKMore data for this Ligand-Target Pair
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182010(7-(pyridin-2-yl)-N-(2,4,6-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50:  212nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair