TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
University Walk
Curated by ChEMBL
University Walk
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Antagonist activity at human recombinant GLUK6 expressed in HEK293 cells assessed as inhibition of glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.09E+3nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibresMore data for this Ligand-Target Pair
Affinity DataKd: 3.94E+3nMAssay Description:Displacement of [3H]S-glutamate from rat GluR5 S1S2 ligand binding core expressed in Escherichia coli (DE3)More data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Antagonism on GLUK5 containing kainate induced deploarization of isolated neonatal rat dorsal root C-fibersMore data for this Ligand-Target Pair