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Found 1 Enz. Inhib. hit(s) for PDB: 2G1O
TargetRenin(Homo sapiens (Human))
Pfizer

LigandPNGBDBM18039(6-ethyl-5-[9-(3-methoxypropyl)-9H-carbazol-2-yl]py...)
Affinity DataIC50:  173nMpH: 7.4 T: 2°CAssay Description:The renin assay utilized a tandem Green Flourescent Protein (tGFP) substrate that was hydrolyzed by human rennin. The tGFP substrate contained a nine...More data for this Ligand-Target Pair