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Found 2 Enz. Inhib. hit(s) for PDB: 2HHA
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM11658((2S,3S)-2-amino-3-[3-(4-methanesulfonylphenyl)-1,2...)
Affinity DataIC50:  122nMAssay Description:Inhibition of human recombinant DPP4 expressed in insect cellMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM11658((2S,3S)-2-amino-3-[3-(4-methanesulfonylphenyl)-1,2...)
Affinity DataIC50:  122nMpH: 7.5 T: 2°CAssay Description:The enzyme activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 360 nm and m...More data for this Ligand-Target Pair