Affinity DataKi: 9.14E+5nMAssay Description:Inhibition of JMJD2EMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMpH: 7.5 T: 2°CAssay Description:A coupled-assay for JMJD2E activity employing formaldehyde dehydrogenase (FDH) from Pseudomonas putida was developed. Formaldehyde release by demethy...More data for this Ligand-Target Pair
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of KDM4E (unknown origin)More data for this Ligand-Target Pair