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Found 1 Enz. Inhib. hit(s) for PDB: 2XJ1
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

LigandPNGBDBM28397((2E)-3-(3-{6-[(4-aminocyclohexyl)amino]pyrazin-2-y...)
Affinity DataIC50:  13nMpH: 7.5 T: 2°CAssay Description:The activity of Pim kinase was measured in a homogeneous luciferase assay using GST-Pim, biotinylated peptide substrate and a luciferin-luciferase de...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed