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Found 3 Enz. Inhib. hit(s) for PDB: 3BYO
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50374608(CHEMBL410295)
Affinity DataIC50:  7nMAssay Description:Inhibition of Lck by HTRF assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50374608(CHEMBL410295)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human T-cell receptor zeta chain phosphorylation in Jurkat cellsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50080265(2-Amino-3-(4-phosphonooxy-phenyl)-propionic acid |...)
Affinity DataKd:  4.00E+5nMAssay Description:Binding affinity against Lck SH2 domainMore data for this Ligand-Target Pair