TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Displacement of [3H2]nTZD3 from GST-tagged human recombinant PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Activation of human PPARgamma-dependent transcription expressed in human MCF7 cells assessed as induction of PPRE-reporter gene expression after 24 h...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Wake Forest University
Curated by ChEMBL
Wake Forest University
Curated by ChEMBL
Affinity DataEC50: 45nMAssay Description:Activation of PPARgammaMore data for this Ligand-Target Pair