Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) for PDB: 3SMR
TargetWD repeat-containing protein 5(Homo sapiens (Human))
Entremed

Curated by ChEMBL
LigandPNGBDBM50428254(CHEMBL1609857)
Affinity DataKd:  6.90E+3nMAssay Description:Displacement of N-terminal isothiocyanate-fluorescein-labeled H3(ARTKQTARKSTGGKA) peptide from human WDR5 expressed in Escherichia coli BL21(DE3) by ...More data for this Ligand-Target Pair
TargetWD repeat-containing protein 5(Homo sapiens (Human))
Entremed

Curated by ChEMBL
LigandPNGBDBM50428254(CHEMBL1609857)
Affinity DataKd:  7.00E+3nMAssay Description:Displacement of N-terminal FITC-labeled GSARAEVHLRKS from WDR5 (1 to 334 residues) (unknown origin) expressed in baculovirus infected Sf9 insect cell...More data for this Ligand-Target Pair
TargetWD repeat-containing protein 5(Homo sapiens (Human))
Entremed

Curated by ChEMBL
LigandPNGBDBM50428254(CHEMBL1609857)
Affinity DataKd:  7.00E+3nMAssay Description:Displacement of MLL-WIN N-terminal FITC-tagged GSARAEVHLRKS peptide from human WDR5 (1-334) by fluorescence polarization assayMore data for this Ligand-Target Pair