Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) for PDB: 4A9R
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant Chk2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)
Affinity DataIC50:  15nMAssay Description:Inhibition of Chk2Checked by AuthorMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)
Affinity DataIC50:  15nMAssay Description:Inhibition of recombinant human Chk2 kinaseMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)
Affinity DataIC50:  15nMAssay Description:Inhibition of Chk2Checked by AuthorMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)
Affinity DataIC50:  16nMAssay Description:Inhibition of chk2 kinaseMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant human Chk2 kinaseMore data for this Ligand-Target Pair
LigandPNGBDBM34064(2-arylbenzimidazole | CHEMBL179583)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:NSC 109555 was diluted in water. All other drugs were dissolved in DMSO, in which case the final DMSO concentration in reactions was 10%, and the con...More data for this Ligand-Target Pair