Found 5 Enz. Inhib. hit(s) for PDB: 4EKL TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 2.60nMAssay Description:iFLiK and HTRF studies were carried out as described in Z. Fang, J. R. Simard, D. Plenker, H. D. Nguyen, T. Phan, P. Wolle, S. Baumeister, D. Rauh, A...More data for this Ligand-Target Pair
3D Structure (crystal)TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 5nMAssay Description:Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt1 expressed in recombinant baculovirus system using fluo...More data for this Ligand-Target Pair
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Array Biopharma
Curated by ChEMBL
Array Biopharma
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt3 expressed in recombinant baculovirus system using fluo...More data for this Ligand-Target Pair
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Array Biopharma
Curated by ChEMBL
Array Biopharma
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt2 expressed in recombinant baculovirus system using fluo...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Technische UniversitÄT Dortmund
US Patent
Technische UniversitÄT Dortmund
US Patent
Affinity DataIC50: 157nMAssay Description:Competitive inhibition of wild-type full-length amino-terminal polyhistidine-tagged human Akt1 expressed in recombinant baculovirus system using fluo...More data for this Ligand-Target Pair
