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Found 2 Enz. Inhib. hit(s) for PDB: 4I9I
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50425969(CHEMBL2314698)
Affinity DataIC50:  2nMAssay Description:Inhibition of N-terminal His6-tagged human TNKS2 (946 to 1162 amino acid residues) after 60 mins by autoparsylation assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50425969(CHEMBL2314698)
Affinity DataIC50:  8nMAssay Description:Inhibition of N-terminal His6-tagged human TNKS1 (1091 to 1325 amino acid residues) after 60 mins by autoparsylation assayMore data for this Ligand-Target Pair