Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) for PDB: 4LZ5
TargetGlutamate receptor 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  559nMAssay Description:Activity against human GLUR2 flip expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  1.91E+3nMAssay Description:Activity against human GLUR2 flop expressed in HEK293 cells assesed as glutamate-stimulated calcium influx by FLIPR assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  1.44E+3nMAssay Description:Inhibition of GluR2 flop expressed in HEK cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  1.66E+3nMAssay Description:Inhibition of GluR3 expressed in HEK cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  5.65E+3nMAssay Description:Inhibition of GluR1 expressed in HEK cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50094024((+/-) Propane-2-sulfonic acid [2-(4'-cyano-bipheny...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at GluR2 receptorMore data for this Ligand-Target Pair