TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences
Curated by ChEMBL
Graduate School Of The Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences
Curated by ChEMBL
Graduate School Of The Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galac...More data for this Ligand-Target Pair