Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 4WLB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50035886(CHEMBL3361065)
Affinity DataIC50:  180nMAssay Description:Displacement of [3H]25-hydroxycholesterol from human RORc-LBD expressed in bacterial expression system after 3 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50035886(CHEMBL3361065)
Affinity DataEC50:  520nMAssay Description:Inverse agonist activity at N-terminal 6xHis-tagged human RORc ligand binding domain expressed in bacterial expression system assessed as inhibition ...More data for this Ligand-Target Pair