Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) for PDB: 5J48
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  163nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351,G182E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  206nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351,G306E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  4.20nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351,G182E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  328nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [5-676,G306E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  370nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [5-676,G306E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  249nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  212nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351,G306E](Homo sapiens (Human))
Baylor College Of Medicine

LigandPNGBDBM65501(8-pCP-cGMP | Cyclic GMP analogs | cGMP)
Affinity DataEC50:  7.70nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair