Found 2 Enz. Inhib. hit(s) for PDB: 5J71 Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
National Institute Of Biological Science
Curated by ChEMBL
National Institute Of Biological Science
Curated by ChEMBL
Affinity DataIC50: 195nMAssay Description:Inhibition of N-terminal His6-SUMO tagged recombinant human PDK2 using [32P]-gamma-ATP assessed as decrease in incorporation of radioactivity into E1...More data for this Ligand-Target Pair
3D Structure (crystal)Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
National Institute Of Biological Science
Curated by ChEMBL
National Institute Of Biological Science
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding affinity to N-terminal His6-SUMO tagged recombinant human PDK2 by isothermal titration calorimetryMore data for this Ligand-Target Pair
