Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) for PDB: 5ZSA
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50330063(1-(4-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  528nMAssay Description:Agonist activity at human TLR7 transfected in HEK reporter cells assessed as NFkappaB induction by specific secreted alkaline phosphatease gene assayMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50330063(1-(4-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human TLR7 expressed in HEK-Blue-7 cells assessed as increase in NFkappaB activation by sAP assayMore data for this Ligand-Target Pair