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Found 4 Enz. Inhib. hit(s) for PDB: 1M0B
TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

LigandPNGBDBM17351((4S)-4-[(2S)-2-{[(3S)-3-{[(tert-butoxy)carbonyl]am...)
Affinity DataKi:  1.5nMpH: 4.7Assay Description:Inhibition constants were determined by a spectrophotometric assay with the chromogenic peptide substrate.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM17351((4S)-4-[(2S)-2-{[(3S)-3-{[(tert-butoxy)carbonyl]am...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of wild type HIV1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM17351((4S)-4-[(2S)-2-{[(3S)-3-{[(tert-butoxy)carbonyl]am...)
Affinity DataKi:  4.10nMAssay Description:Inhibition of HIV1 protease I8 mutantMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [501-599,A572V,V583T,I585V](Human immunodeficiency virus type 1)
Academy Of Sciences Of The Czech Republic

LigandPNGBDBM17351((4S)-4-[(2S)-2-{[(3S)-3-{[(tert-butoxy)carbonyl]am...)
Affinity DataKi:  4.10nMpH: 4.7Assay Description:Inhibition constants were determined by a spectrophotometric assay with the chromogenic peptide substrate.More data for this Ligand-Target Pair