Affinity DataIC50: 5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of porcine brain GSK3beta using YRRAAVPPSPSLSRHSSPHQSpEDEEE as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to GSK3alphaChecked by AuthorMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)
Curated by ChEMBL
Jamia Hamdard (Hamdard University)
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)
Curated by ChEMBL
Jamia Hamdard (Hamdard University)
Curated by ChEMBL
Affinity DataEC50: >3.00E+6nMAssay Description:Effective concentration of compound against glycogen synthase kinase-3 in HEK293 cellsMore data for this Ligand-Target Pair