Found 3 Enz. Inhib. hit(s) for PDB: 2A5U TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of California San Francisco
University Of California San Francisco
Affinity DataIC50: 8nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
3D Structure (crystal)TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of California San Francisco
University Of California San Francisco
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged PI3K-gamma (39 to 1102 residues) expressed n baculovirus infected TN5 cells using phosphatidyli...More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
University Of California San Francisco
University Of California San Francisco
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant GST-tagged PI3Kgamma incubated for 180 mins using [33P]gamma-ATP by scintillation proximity assayMore data for this Ligand-Target Pair
