Found 3 Enz. Inhib. hit(s) for PDB: 2C3J TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 725nMAssay Description:Inhibition of human CHK1 using STK1 as substrate after 10 mins by HTRF assayMore data for this Ligand-Target Pair
3D Structure (crystal)TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 725nMAssay Description:Inhibition of CHK1 (unknown origin) using polypeptide substrate after 40 mins in presence of [gamma-33P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Chk1Checked by AuthorMore data for this Ligand-Target Pair
