Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) for PDB: 2OPB
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50151343((+)-3-(fluoromethyl)-7-(thiomorpholinosulfonyl)-1,...)
Affinity DataKi:  315nMAssay Description:Inhibition of wild type human PNMTMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50163110((3R)-3-(FLUOROMETHYL)-7-(THIOMORPHOLIN-4-YLSULFONY...)
Affinity DataKi:  610nMAssay Description:In vitro binding affinity against recombinant human Phenylethanolamine N-methyltransferase expressed in E. coli using [methyl-3H]-AdoMetMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50151343((+)-3-(fluoromethyl)-7-(thiomorpholinosulfonyl)-1,...)
Affinity DataKi:  1.20E+3nMAssay Description:In vitro binding affinity against recombinant human Phenylethanolamine N-methyltransferase expressed in E. coli using [methyl-3H]-AdoMetMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50151343((+)-3-(fluoromethyl)-7-(thiomorpholinosulfonyl)-1,...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of [3H]-methyl-AdoMet binding to human phenylethnolamine N-methyltransferase expressed in E. coli BL21More data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50151343((+)-3-(fluoromethyl)-7-(thiomorpholinosulfonyl)-1,...)
Affinity DataKi:  1.20E+3nMAssay Description:In vitro binding affinity against human phenylethanolamine N-MethyltransferaseMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition constant was evaluated against PNMTMore data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition constant was evaluated against PNMTMore data for this Ligand-Target Pair