Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) for PDB: 2Q59
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157933(2-{2-[1-(4-Methoxy-benzoyl)-2-methyl-5-trifluorome...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50157936((2S)-2-(2-{[1-(4-METHOXYBENZOYL)-2-METHYL-5-(TRIFL...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of human Peroxisome proliferator activated receptor gammaMore data for this Ligand-Target Pair