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Found 3 Enz. Inhib. hit(s) for PDB: 3IX3
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  31nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasRMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR expressed in Escherichia coli JLD271 harboring LasR expression plasmid pJN105L and lasI-lacZ transcri...More data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Rowan University

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  7nMAssay Description:Agonist activity at Pseudomonas aeruginosa LasR cognate receptor expressed in Escherichia coli harboring pKDT17 assessed as activation of lasB expres...More data for this Ligand-Target Pair