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Found 3 Enz. Inhib. hit(s) for PDB: 3KF4
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50244569(AP24283 | CHEMBL510893 | N-(4-(dimethylphosphoryl)...)
Affinity DataIC50: <0.460nMAssay Description:Inhibition of Abl kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50244569(AP24283 | CHEMBL510893 | N-(4-(dimethylphosphoryl)...)
Affinity DataIC50: <0.5nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
Ariad Pharmaceuticals

LigandPNGBDBM50244569(AP24283 | CHEMBL510893 | N-(4-(dimethylphosphoryl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair