TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of wild type ROS1 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Inhibition of ROS1 L2026M mutant (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataKi: 330nMAssay Description:Inhibition of ROS1 G2032R mutant (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of ROS1 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of ROS1 (unknown origin) using peptide as substrate after 60 mins by HTRF assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged ROS1 cytoplasmic domain (1883 to 2347 residues) expressed in baculovirus expression system usin...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataIC50: 199nMAssay Description:Inhibition of ROS1 (unknown origin) incubated for 20 mins followed by [33P]ATP addition measured after 120 mins by HotSpot assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human N-terminal GST-tagged ROS cytoplasmic domain (1883 to 2347 residues) expressed in baculovirus expression system after 1 hr by mob...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Taibah University
Curated by ChEMBL
Taibah University
Curated by ChEMBL
Affinity DataKd: 4.10nMAssay Description:Binding constant for ROS1 kinase domainMore data for this Ligand-Target Pair