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Found 4 Enz. Inhib. hit(s) for PDB: 3ZYA
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
University Of Zagreb

Curated by ChEMBL
LigandPNGBDBM50241112(2-(2-Amino-phenylamino)-10,11-dihydro-dibenzo[a,d]...)
Affinity DataIC50:  50nMAssay Description:Inhibition of MAPK p38 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50241112(2-(2-Amino-phenylamino)-10,11-dihydro-dibenzo[a,d]...)
Affinity DataIC50:  50nMAssay Description:Inhibition of MAP kinase p38alpha assessed as phosphorylation of ATF-2More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50241112(2-(2-Amino-phenylamino)-10,11-dihydro-dibenzo[a,d]...)
Affinity DataIC50:  100nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) by cell-free enzyme immunosorbent assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50241112(2-(2-Amino-phenylamino)-10,11-dihydro-dibenzo[a,d]...)
Affinity DataIC50:  104nMAssay Description:Inhibition of p38 alphaMore data for this Ligand-Target Pair