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Found 5 Enz. Inhib. hit(s) for PDB: 4AJH
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86124(LDHA Inhibitor, 20)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86126(LDHA Inhibitor, 22)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86126(LDHA Inhibitor, 22)
Affinity DataKd:  7.70E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86124(LDHA Inhibitor, 20)
Affinity DataKd:  4.70E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86124(LDHA Inhibitor, 20)
Affinity DataKd:  2.10E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair