Affinity DataIC50: 5nMAssay Description:Inhibition of CDK8/CCNC (unknown origin) using RBER-IRStide as substrate in presence of [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 19(Homo sapiens (Human))
University Of South Australia
Curated by ChEMBL
University Of South Australia
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK19 (unknown origin) in presence of [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of CDK8 (unknown origin) assessed as reduction in RNAP2 C-terminal domain phosphorylationMore data for this Ligand-Target Pair