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Found 2 Enz. Inhib. hit(s) for PDB: 4HLF
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University Of Oulu

Curated by ChEMBL
LigandPNGBDBM50077325(2-(3,4-Dihydroxy-phenyl)-7-hydroxy-chromen-4-one |...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human 6XHis-tagged TNKS1 SAM-ART domain (1030 to 1317 amino acid residues) by fluorescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University Of Oulu

Curated by ChEMBL
LigandPNGBDBM50077325(2-(3,4-Dihydroxy-phenyl)-7-hydroxy-chromen-4-one |...)
Affinity DataIC50:  870nMAssay Description:Inhibition of human 6XHis-tagged TNKS2 ART domain (946 to 1161 amino acid residues) expressed in Escherichia coli Rosetta2 (DE3) by fluorescence assa...More data for this Ligand-Target Pair