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Found 2 Enz. Inhib. hit(s) for PDB: 4JLM
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440155(CHEMBL2426598)
Affinity DataIC50:  7nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440155(CHEMBL2426598)
Affinity DataIC50:  30nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair