Affinity DataKd: 350nMAssay Description:Binding affinity to GluA2-LBD-L483Y-N754S complex (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Positive allosteric modulation of GluA2 receptor in rat embryonic cortex neuron assessed as increase of AMPA-induced membrane depolarization by fluor...More data for this Ligand-Target Pair
Affinity DataEC50: 813nMAssay Description:Positive allosteric modulation of GluA2 (Q) flop isoform (unknown origin) expressed in HEK293 cells assessed as potentiation of glutamate-evoked calc...More data for this Ligand-Target Pair
Affinity DataEC50: 810nMAssay Description:Positive allosteric modulation of GluA2 (Q) flop isoform (unknown origin) expressed in HEK293 cells assessed as potentiation of glutamate-evoked calc...More data for this Ligand-Target Pair