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Found 1 Enz. Inhib. hit(s) for PDB: 4XUH
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Vanderbilt University Center For Structural Biology

Curated by ChEMBL
LigandPNGBDBM50110164((Z)-2-(3-(4-(methylthio)benzylidene)-6-fluoro-2-me...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at PPARgamma expressed in human HCA7 cells assessed as induction of peroxisome proliferator response element after 12 hrs by lucifer...More data for this Ligand-Target Pair