Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) for PDB: 5LUU
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50207718(CHEMBL3959972)
Affinity DataKd:  3.13E+4nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using 1% DMSO by SPR assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50207718(CHEMBL3959972)
Affinity DataKd:  8.63E+3nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using methanol by SPR assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50207718(CHEMBL3959972)
Affinity DataKd:  1.74E+4nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using 0.5% DMSO by SPR assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM50207718(CHEMBL3959972)
Affinity DataKd:  9.70E+4nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using 3% DMSO by SPR assayMore data for this Ligand-Target Pair