Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) for PDB: 5LWE
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataKi:  1.10nMAssay Description:Antagonist activity at CCR9 receptor in human MOLT4 cells assessed as inhibition of CCL25-induced increase in intracellular calcium level preincubate...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataKi:  3.70nMAssay Description:Antagonist activity at CCR9A receptor (unknown origin) overexpressed in human MOLT4 cells assessed as inhibition of CCL25-induced increase in intrace...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataKi:  10nMAssay Description:Antagonist activity at CCR9 receptor in human MOLT4 cells assessed as inhibition of CCl25-mediated cell migration preincubated for 30 mins followed C...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataIC50:  2.80nMAssay Description:Antagonist activity at CCR9 assessed as inhibition of CCL25-induced chemotaxis by cell based assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at CCR9 (unknown origin) assessed as inhibition of TECK-stimulated calcium mobilization preincubated for 10 mins followed by agon...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataIC50:  6nMAssay Description:Binding affinity to CCR9More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Norgine

Curated by ChEMBL
LigandPNGBDBM50398334(CHEMBL2178578)
Affinity DataIC50:  539nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by serum chemotaxis assayMore data for this Ligand-Target Pair