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Found 1 Enz. Inhib. hit(s) for PDB: 5MRH
TargetSortilin(Homo sapiens (Human))
Aarhus University

Curated by ChEMBL
LigandPNGBDBM50249496(CHEMBL4081301)
Affinity DataIC50:  6.31E+4nMAssay Description:Displacement of [3H]-neurotensin from human His6-tagged sortilin pretreated for 30 mins followed by [3H]-neurotensin addition after 6 hrs measured fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB