Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) for PDB: 5TLU
TargetEstrogen receptor(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50309555(17alpha-(4-Aminophenyl)ethynyl-estra-1,3,5(10)-tri...)
Affinity DataEC50:  10nMAssay Description:Estrogenic activity at ERalpha in human Ishikawa cells assessed as stimulation of alkaline phosphatase activity after 4 days by microplate scanning s...More data for this Ligand-Target Pair