Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) for PDB: 5Z8G
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405922(CHEMBL4167407)
Affinity DataIC50:  3.22E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair