Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) for PDB: 5Z90
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50238042(CHEMBL4073350)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of human BRD4-BD1 (49 to 170 residues) expressed in Escherichia coli BL21(DE3) using N-C:SGRG-K(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHRKVGG-K...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Nanchang University

Curated by ChEMBL
LigandPNGBDBM50238042(CHEMBL4073350)
Affinity DataIC50:  6.83E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair