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Found 14 Enz. Inhib. hit(s) with all data for entry = 50008629
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50075437(2,4,5-Trifluoro-6-nitro-3-((2E,6E)-3,7,11-trimethy...)
Affinity DataIC50:  6.30E+3nMAssay Description:In vitro inhibition of rat brain cytosol farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075437(2,4,5-Trifluoro-6-nitro-3-((2E,6E)-3,7,11-trimethy...)
Affinity DataIC50:  1.25E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075439(3-Benzyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMB...)
Affinity DataIC50:  5.80E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075440(2,4,5-Trifluoro-3-(4-isopropenyl-cyclohex-1-enylme...)
Affinity DataIC50:  8.50E+4nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075443(3-Dodecyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50075443(3-Dodecyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEM...)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50075440(2,4,5-Trifluoro-3-(4-isopropenyl-cyclohex-1-enylme...)
Affinity DataIC50:  1.20E+5nMAssay Description:In vitro antagonistic activity against endothelin B receptor in isolated rabbit jugularis veinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50075441(2,4,5-Trifluoro-3-(naphthalen-2-ylmethoxy)-6-nitro...)
Affinity DataIC50:  2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50075438(3-(Biphenyl-4-ylmethoxy)-2,4,5-trifluoro-6-nitro-p...)
Affinity DataIC50:  2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50075439(3-Benzyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMB...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50075442(3-Allyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMBL...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro antagonistic activity against endothelin A receptor in isolated rat aortic ringsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075441(2,4,5-Trifluoro-3-(naphthalen-2-ylmethoxy)-6-nitro...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075438(3-(Biphenyl-4-ylmethoxy)-2,4,5-trifluoro-6-nitro-p...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50075442(3-Allyloxy-2,4,5-trifluoro-6-nitro-phenol | CHEMBL...)
Affinity DataIC50: >2.00E+5nMAssay Description:In vitro inhibition of rat brain cytosol Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed