Compile Data Set for Download or QSAR
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Found 35 Enz. Inhib. hit(s) with all data for entry = 50009040
TargetD(4) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079644(2-[4-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity of compound towards human cloned Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079645(2-{4-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity of compound towards human cloned Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079642(2-[5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  9.30nMAssay Description:Binding affinity of compound towards human cloned Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079646(2-{5-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  11nMAssay Description:Binding affinity of compound towards human cloned Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  16nMAssay Description:Binding affinity of compound towards human cloned Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  28nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2S stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  39nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2L stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(4) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079641(2-{3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  125nMAssay Description:Binding affinity of compound towards human cloned Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079643(2-[3-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  160nMAssay Description:Binding affinity of compound towards human cloned Dopamine receptor D4.4 expressed in CHO cells using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  420nMAssay Description:Ability of the compound to displace D1 selective radioligand [3H]-SCH- 23390 in bovine striatal membrane preparations was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  960nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human D3 dopamine receptor stably expressed in Chinese hamster ovary (CHO) cells w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079644(2-[4-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  975nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2S stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079644(2-[4-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  1.85E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2L stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079644(2-[4-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  2.35E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human D3 dopamine receptor stably expressed in Chinese hamster ovary (CHO) cells w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079643(2-[3-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  4.00E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2L stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079642(2-[5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  5.25E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human D3 dopamine receptor stably expressed in Chinese hamster ovary (CHO) cells w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079645(2-{4-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  5.30E+3nMAssay Description:Ability of the compound to displace D1 selective radioligand [3H]-SCH- 23390 in bovine striatal membrane preparations was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079643(2-[3-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  6.95E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human D3 dopamine receptor stably expressed in Chinese hamster ovary (CHO) cells w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079645(2-{4-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  6.95E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human D3 dopamine receptor stably expressed in Chinese hamster ovary (CHO) cells w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079644(2-[4-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  7.20E+3nMAssay Description:Ability of the compound to displace D1 selective radioligand [3H]-SCH- 23390 in bovine striatal membrane preparations was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079645(2-{4-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  7.35E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2L stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079641(2-{3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  7.60E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human D3 dopamine receptor stably expressed in Chinese hamster ovary (CHO) cells w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079641(2-{3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  8.95E+3nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2L stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079645(2-{4-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  1.03E+4nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2S stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079643(2-[3-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  1.28E+4nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2S stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079641(2-{3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  1.35E+4nMAssay Description:Ability of the compound to displace D1 selective radioligand [3H]-SCH- 23390 in bovine striatal membrane preparations was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079641(2-{3-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  1.50E+4nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2S stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079643(2-[3-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  2.20E+4nMAssay Description:Ability of the compound to displace D1 selective radioligand [3H]-SCH- 23390 in bovine striatal membrane preparations was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079646(2-{5-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  3.10E+4nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human D3 dopamine receptor stably expressed in Chinese hamster ovary (CHO) cells w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079646(2-{5-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  3.95E+4nMAssay Description:Ability of the compound to displace D1 selective radioligand [3H]-SCH- 23390 in bovine striatal membrane preparations was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079646(2-{5-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  4.85E+4nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2L stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(BOVINE)
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079642(2-[5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi:  5.80E+4nMAssay Description:Ability of the compound to displace D1 selective radioligand [3H]-SCH- 23390 in bovine striatal membrane preparations was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079646(2-{5-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-1H...)
Affinity DataKi:  5.90E+4nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2S stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079642(2-[5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi: >1.00E+5nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2L stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
UniversitäT Erlangen - NüRnberg

Curated by ChEMBL
LigandPNGBDBM50079642(2-[5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrol-2-y...)
Affinity DataKi: >1.00E+5nMAssay Description:Ability of the compound to displace [3H]-spiperone from the cloned human Dopamine receptor D2S stably expressed in Chinese hamster ovary (CHO) cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed