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Found 10 Enz. Inhib. hit(s) with all data for entry = 50035019
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081427((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081428((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081429((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  2.90E+4nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081429((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  6.30E+4nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081428((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  1.02E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081426((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  1.32E+5nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081427((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50:  1.72E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081426((4R,4aS)-4,8-Dihydroxy-6-methyl-9-oxo-4,9-dihydro-...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2(Drosophila melanogaster)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081431(7,16-dihydroxy-5,14-dimethyl-(1S,13S,16R)-2-oxa-14...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibitory activity against topoisomerase II (Topo II) by using decatenation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Mus musculus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50081431(7,16-dihydroxy-5,14-dimethyl-(1S,13S,16R)-2-oxa-14...)
Affinity DataIC50: >3.00E+5nMAssay Description:In vitro inhibitory activity against topoisomerase I (Topo I) by using relaxation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed