Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50009517
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50068366(CHEMBL93403 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  0.0400nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084496(4-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi:  4nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084486(CHEMBL92713 | N-{3-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  5.40nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  5.60nMAssay Description:In vitro binding affinity towards Dopamine receptor D2L, using [3H]-spiroperidol radioligand in Sf9 baculovirus expression.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084489(2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-7...)
Affinity DataKi:  11nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084481(5-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi:  21nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084493(CHEMBL96462 | {2-[4-(4-Chloro-phenyl)-piperazin-1-...)
Affinity DataKi:  23nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084494(CHEMBL315879 | N-{4-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  30nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084481(5-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi:  37nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084487(2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-5...)
Affinity DataKi:  42nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084483(3-[4-(4-Chloro-phenyl)-piperazin-1-yl]-N-(3-methox...)
Affinity DataKi:  42nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084482(6-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi:  45nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084495(CHEMBL328283 | {2-[4-(4-Chloro-phenyl)-piperazin-1...)
Affinity DataKi:  46nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084485(1-(4-Chloro-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetrah...)
Affinity DataKi:  105nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084489(2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-7...)
Affinity DataKi:  141nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50068366(CHEMBL93403 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  147nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084488(CHEMBL92411 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  180nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084496(4-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi:  183nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084492(1-(4-Chloro-phenyl)-4-[4-(3-methoxy-phenyl)-butyl]...)
Affinity DataKi:  204nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084484(CHEMBL94265 | N-{5-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  241nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084495(CHEMBL328283 | {2-[4-(4-Chloro-phenyl)-piperazin-1...)
Affinity DataKi:  262nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084482(6-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi:  280nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084483(3-[4-(4-Chloro-phenyl)-piperazin-1-yl]-N-(3-methox...)
Affinity DataKi:  282nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084491(1-(4-Chloro-phenyl)-4-[3-(7-methoxy-1,2,3,4-tetrah...)
Affinity DataKi:  391nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084494(CHEMBL315879 | N-{4-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi:  397nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084485(1-(4-Chloro-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetrah...)
Affinity DataKi:  416nMAssay Description:In vitro binding affinity at human Dopamine receptor D4.4 by [3H]-YM-09151-2 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  443nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine receptor 1A receptor by using [3H]-8-OH-DPAT in rat hippocampal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084487(2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-5...)
Affinity DataKi:  451nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084492(1-(4-Chloro-phenyl)-4-[4-(3-methoxy-phenyl)-butyl]...)
Affinity DataKi:  514nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084491(1-(4-Chloro-phenyl)-4-[3-(7-methoxy-1,2,3,4-tetrah...)
Affinity DataKi:  708nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084493(CHEMBL96462 | {2-[4-(4-Chloro-phenyl)-piperazin-1-...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084482(6-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084481(5-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084488(CHEMBL92411 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084484(CHEMBL94265 | N-{5-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084484(CHEMBL94265 | N-{5-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084486(CHEMBL92713 | N-{3-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084488(CHEMBL92411 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084495(CHEMBL328283 | {2-[4-(4-Chloro-phenyl)-piperazin-1...)
Affinity DataKi: >850nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084483(3-[4-(4-Chloro-phenyl)-piperazin-1-yl]-N-(3-methox...)
Affinity DataKi:  859nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine receptor 1A receptor in rat hippocampal membranes by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  876nMAssay Description:In vitro binding affinity towards Dopamine receptor D2L, using [3H]-spiroperidol radioligand in Sf9 baculovirus expression.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084491(1-(4-Chloro-phenyl)-4-[3-(7-methoxy-1,2,3,4-tetrah...)
Affinity DataKi:  980nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50068366(CHEMBL93403 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  1.90E+3nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084494(CHEMBL315879 | N-{4-[4-(4-Chloro-phenyl)-piperazin...)
Affinity DataKi:  2.35E+3nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universitá

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  2.39E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine receptor 1A receptor by using [3H]-8-OH-DPAT in rat hippocampal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084496(4-[4-(4-Chloro-phenyl)-piperazin-1-yl]-1-(3-methox...)
Affinity DataKi:  2.55E+3nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084492(1-(4-Chloro-phenyl)-4-[4-(3-methoxy-phenyl)-butyl]...)
Affinity DataKi:  2.74E+3nMAssay Description:In vitro binding affinity at human Dopamine receptor D2 (long) by [3H]-spiroperidol displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universitá

Curated by ChEMBL
LigandPNGBDBM50084487(2-{2-[4-(4-Chloro-phenyl)-piperazin-1-yl]-ethyl}-5...)
Affinity DataKi:  3.17E+3nMAssay Description:In vitro binding affinity towards human Dopamine receptor D2L, using [3H]-spiroperidol radioligand in Sf9 baculovirus expression.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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