Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50009764
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087556((4-Fluoro-butyl)-propyl-[2,5,6-trimethyl-7-(2,4,6-...)
Affinity DataKi:  0.910nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087559(CHEMBL164206 | Cyclopropylmethyl-propyl-[2,5,6-tri...)
Affinity DataKi:  2.30nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50074501(Butyl-ethyl-[2,5,6-trimethyl-7-(2,4,6-trimethyl-ph...)
Affinity DataKi:  2.5nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087560(CHEMBL348967 | Ethyl-(4-fluoro-butyl)-[2,5,6-trime...)
Affinity DataKi:  3.5nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087561(Butyl-(4-fluoro-butyl)-[2,5,6-trimethyl-7-(2,4,6-t...)
Affinity DataKi:  10nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087557(CHEMBL164042 | Cyclopropylmethyl-(3-fluoro-propyl)...)
Affinity DataKi:  30nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50087558(4-[4-(2-Fluoro-ethyl)-piperazin-1-yl]-2,5,6-trimet...)
Affinity DataKi: >1.00E+3nMAssay Description:Compound was tested in vitro for its ability to displace [125 I]Tyr-sauvagine from corticotropin-releasing hormone type 1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed