Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50009796
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087851(CHEMBL384518 | LysProSerProAspArgPheTyrGlyLeuMet)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  0.600nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087850(CHEMBL415159 | TyrLysSerAspSerPheTyrGlyLeuMet)
Affinity DataEC50:  14nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087850(CHEMBL415159 | TyrLysSerAspSerPheTyrGlyLeuMet)
Affinity DataEC50:  14nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087852(CHEMBL263185 | His-Asn-Pro-Ala-Ser-Phe-Ile-Gly-Leu...)
Affinity DataEC50:  13.5nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087852(CHEMBL263185 | His-Asn-Pro-Ala-Ser-Phe-Ile-Gly-Leu...)
Affinity DataEC50:  14nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center

Curated by ChEMBL
LigandPNGBDBM50087851(CHEMBL384518 | LysProSerProAspArgPheTyrGlyLeuMet)
Affinity DataEC50:  0.600nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed