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Found 233 Enz. Inhib. hit(s) with all data for entry = 50036926
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50037996(1-[N-(naphthalen-2-ylsulfonyl)glycyl-4-carbamimido...)
Affinity DataKi:  6.5nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087898(1-(3-Phenyl-2-(N-Toluene-4-sulfonyl)ureido-propion...)
Affinity DataKi:  10nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087941(CHEMBL301811 | N-{4-[(N-Guanidino)-sulfamoyl]-phen...)
Affinity DataKi:  10nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087955(CHEMBL52917 | [2-(2-{4-[(N-Guanidino)-sulfamoyl]-p...)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087983(CHEMBL298925 | N-[4-(Diaminomethylene-sulfamoyl)-p...)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087903((1-Benzyl-2-{2-[4-(diaminomethylene-sulfamoyl)-phe...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087962(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087888(CHEMBL53802 | N-{4-[(N-Guanidino)-sulfamoyl]-pheny...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087960(CHEMBL299617 | {1-Cyclohexylmethyl-2-[2-(3-guanidi...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087907(CHEMBL298127 | N-[4-(Diaminomethylene-sulfamoyl)-p...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087963(CHEMBL300666 | [2-(2-{4-[(Amino-methoxy-methylene)...)
Affinity DataKi:  16nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087998(CHEMBL50191 | N-[4-(Diaminomethylene-sulfamoyl)-ph...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087954(1-(3-Phenyl-2-(N-Toluene-4-sulfonyl)ureido-propion...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087994(CHEMBL50689 | N-{4-[(Amino-methoxy-methylene)-sulf...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087965(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087967(CHEMBL50296 | N-{4-[(Amino-methoxy-methylene)-sulf...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087902(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087959(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087953(CHEMBL51635 | {1-[4-(Diaminomethylene-sulfamoyl)-p...)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087901(CHEMBL50590 | N-{4-[(N-Guanidino)-sulfamoyl]-pheny...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087973(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087886((1-{4-[(N-Guanidino)-sulfamoyl]-phenylcarbamoyl}-2...)
Affinity DataKi:  50nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087930(CHEMBL296177 | {1-[4-(Diaminomethylene-sulfamoyl)-...)
Affinity DataKi:  54nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087921(CHEMBL53464 | N-{4-[(Amino-methoxy-methylene)-sulf...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087969((1-{4-[(Amino-methoxy-methylene)-sulfamoyl]-phenyl...)
Affinity DataKi:  62nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087923(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  63nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087912(CHEMBL432326 | N''-[(3-aminophenyl)sulfonyl]carbon...)
Affinity DataKi:  88nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087925(CHEMBL300873 | N''-[(4-aminophenyl)sulfonyl]carbon...)
Affinity DataKi:  91nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50027795(1N-amino(imino)methyl-4-amino-1-benzenesulfonamide...)
Affinity DataKi:  95nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087884(3-Amino-N-(amino-methoxy-methylene)-4-methoxy-benz...)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087885(4-{[2-(diaminomethylene)hydrazino]sulfonyl}benzoic...)
Affinity DataKi:  97nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087897(CHEMBL300708 | N''-[(3,5-dichloro-2-hydroxyphenyl)...)
Affinity DataKi:  98nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087966(3-Amino-N-(amino-methoxy-methylene)-benzenesulfona...)
Affinity DataKi:  99nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087993(3-Amino-N-diaminomethylene-4-methoxy-benzenesulfon...)
Affinity DataKi:  103nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087894(4-(Diaminomethylene-sulfamoyl)-benzoic acid | CHEM...)
Affinity DataKi:  104nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087991(4-Amino-N-(amino-methoxy-methylene)-benzenesulfona...)
Affinity DataKi:  106nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087951(3-Amino-N-diaminomethylene-benzenesulfonamide | CH...)
Affinity DataKi:  107nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087890(3-{[2-(diaminomethylene)hydrazino]sulfonyl}benzoic...)
Affinity DataKi:  112nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087945(5-Dimethylamino-naphthalene-1-sulfonic acid diamin...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087948(3-(Diaminomethylene-sulfamoyl)-benzoic acid | CHEM...)
Affinity DataKi:  121nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087940(CHEMBL54250 | N''-[(pentafluorophenyl)sulfonyl]car...)
Affinity DataKi:  123nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087986(CHEMBL51392 | N''-(1-naphthylsulfonyl)carbonohydra...)
Affinity DataKi:  125nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087976(CHEMBL301987 | N''-(2-naphthylsulfonyl)carbonohydr...)
Affinity DataKi:  129nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087920(CHEMBL50467 | N''-{[5-(dimethylamino)-1-naphthyl]s...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087947(CHEMBL53960 | Naphthalene-2-sulfonic acid diaminom...)
Affinity DataKi:  132nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087933(4-[(Amino-methoxy-methylene)-sulfamoyl]-benzoic ac...)
Affinity DataKi:  133nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087937(CHEMBL298996 | N-Diaminomethylene-4-(4-dimethylami...)
Affinity DataKi:  134nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087918(CHEMBL52846 | Naphthalene-1-sulfonic acid diaminom...)
Affinity DataKi:  136nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50087932(5-Dimethylamino-naphthalene-1-sulfonic acid amino-...)
Affinity DataKi:  138nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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