Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50036813
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50001107(2-(3,4-Dichloro-phenyl)-1-(5-hydroxy-1-pyrrolidin-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50008888((threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-methyl-pyrr...)
Affinity DataKi:  0.330nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50088377(1-{2-[3-(3,4-Dichloro-phenyl)-2-oxo-tetrahydro-pyr...)
Affinity DataKi:  0.420nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50088379(1-[4-(5,6-Dichloro-indane-1-carbonyl)-thiomorpholi...)
Affinity DataKi:  0.440nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50088375(1-{8-[(2,3-Diphenyl-cycloprop-2-enecarbonyl)-methy...)
Affinity DataKi:  0.640nMAssay Description:Inhibition of [3H]- U-69593 binding in cloned rat Opioid receptor kappa 1 expressed in CHO cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  0.890nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50088380(1-(1-{[2-(3,4-Dichloro-phenyl)-acetyl]-methyl-amin...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50088374(1-{2-[3-(3,4-Dichloro-phenyl)-2-oxo-pyrrolidin-1-y...)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]EKC binding to Opioid receptor kappa 1 in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed