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PubMed code 10937714

Compile data set for download or QSAR
Found 19 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090395
PNG
(CHEMBL42762 | N-(6-Hydroxy-1-pyridin-3-ylmethyl-1,...)
Show SMILES Oc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CCC(CC1)n1c2ccccc2[nH]c1=O
Show InChI InChI=1S/C30H33N5O3/c36-23-8-9-24-21(17-23)7-10-26(25(24)16-20-4-3-13-31-18-20)32-29(37)19-34-14-11-22(12-15-34)35-28-6-2-1-5-27(28)33-30(35)38/h1-6,8-9,13,17-18,22,25-26,36H,7,10-12,14-16,19H2,(H,32,37)(H,33,38)
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n/an/a 6n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090398
PNG
(CHEMBL45199 | [4-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Show SMILES CC(C)(C)OC(=O)NC[C@H]1CC[C@@H](CC1)C(=O)NC1CCc2cc(F)ccc2C1Cc1cccnc1
Show InChI InChI=1S/C29H38FN3O3/c1-29(2,3)36-28(35)32-18-19-6-8-21(9-7-19)27(34)33-26-13-10-22-16-23(30)11-12-24(22)25(26)15-20-5-4-14-31-17-20/h4-5,11-12,14,16-17,19,21,25-26H,6-10,13,15,18H2,1-3H3,(H,32,35)(H,33,34)/t19-,21-,25?,26?
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n/an/a 16n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090403
PNG
(CHEMBL43659 | {(S)-1-[(6-Fluoro-1-pyridin-3-ylmeth...)
Show SMILES CC(C)(C)OC(=O)N[C@H]1CCN(CC(=O)NC2CCc3cc(F)ccc3C2Cc2cccnc2)C1
Show InChI InChI=1S/C27H35FN4O3/c1-27(2,3)35-26(34)30-21-10-12-32(16-21)17-25(33)31-24-9-6-19-14-20(28)7-8-22(19)23(24)13-18-5-4-11-29-15-18/h4-5,7-8,11,14-15,21,23-24H,6,9-10,12-13,16-17H2,1-3H3,(H,30,34)(H,31,33)/t21-,23?,24?/m0/s1
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n/an/a 17n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090390
PNG
(2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperi...)
Show SMILES O=C(CN1CCC(CC1)n1c2ccccc2[nH]c1=O)NC1CCc2ccccc2C1Cc1cccnc1
Show InChI InChI=1S/C30H33N5O2/c36-29(20-34-16-13-23(14-17-34)35-28-10-4-3-9-27(28)33-30(35)37)32-26-12-11-22-7-1-2-8-24(22)25(26)18-21-6-5-15-31-19-21/h1-10,15,19,23,25-26H,11-14,16-18,20H2,(H,32,36)(H,33,37)
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n/an/a 22n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090402
PNG
(CHEMBL296022 | N-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CCC(CC1)n1c2ccccc2[nH]c1=O
Show InChI InChI=1S/C30H32FN5O2/c31-22-8-9-24-21(17-22)7-10-26(25(24)16-20-4-3-13-32-18-20)33-29(37)19-35-14-11-23(12-15-35)36-28-6-2-1-5-27(28)34-30(36)38/h1-6,8-9,13,17-18,23,25-26H,7,10-12,14-16,19H2,(H,33,37)(H,34,38)
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n/an/a 25n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090388
PNG
(CHEMBL42658 | N-{(S)-1-[(6-Fluoro-1-pyridin-3-ylme...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CC[C@@H](C1)NC(=O)c1ccccc1
Show InChI InChI=1S/C29H31FN4O2/c30-23-9-10-25-22(16-23)8-11-27(26(25)15-20-5-4-13-31-17-20)33-28(35)19-34-14-12-24(18-34)32-29(36)21-6-2-1-3-7-21/h1-7,9-10,13,16-17,24,26-27H,8,11-12,14-15,18-19H2,(H,32,36)(H,33,35)/t24-,26?,27?/m0/s1
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n/an/a 26n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090392
PNG
(CHEMBL44886 | N-{1-[(6-Fluoro-1-pyridin-3-ylmethyl...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CCC(CC1)NC(=O)c1ccccc1
Show InChI InChI=1S/C30H33FN4O2/c31-24-9-10-26-23(18-24)8-11-28(27(26)17-21-5-4-14-32-19-21)34-29(36)20-35-15-12-25(13-16-35)33-30(37)22-6-2-1-3-7-22/h1-7,9-10,14,18-19,25,27-28H,8,11-13,15-17,20H2,(H,33,37)(H,34,36)
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n/an/a 28n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090401
PNG
(CHEMBL42031 | {(R)-1-[(6-Fluoro-1-pyridin-3-ylmeth...)
Show SMILES CC(C)(C)OC(=O)N[C@@H]1CCN(CC(=O)NC2CCc3cc(F)ccc3C2Cc2cccnc2)C1
Show InChI InChI=1S/C27H35FN4O3/c1-27(2,3)35-26(34)30-21-10-12-32(16-21)17-25(33)31-24-9-6-19-14-20(28)7-8-22(19)23(24)13-18-5-4-11-29-15-18/h4-5,7-8,11,14-15,21,23-24H,6,9-10,12-13,16-17H2,1-3H3,(H,30,34)(H,31,33)/t21-,23?,24?/m1/s1
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n/an/a 30n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090396
PNG
(CHEMBL44036 | [4-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)[C@H]1CC[C@H](CNC(=O)Oc2ccccc2)CC1
Show InChI InChI=1S/C31H34FN3O3/c32-25-13-14-27-24(18-25)12-15-29(28(27)17-22-5-4-16-33-19-22)35-30(36)23-10-8-21(9-11-23)20-34-31(37)38-26-6-2-1-3-7-26/h1-7,13-14,16,18-19,21,23,28-29H,8-12,15,17,20H2,(H,34,37)(H,35,36)/t21-,23-,28?,29?
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n/an/a 31n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090389
PNG
(CHEMBL288763 | N-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CCC(CC1)NC(=O)Cc1ccccc1
Show InChI InChI=1S/C31H35FN4O2/c32-25-9-10-27-24(19-25)8-11-29(28(27)17-23-7-4-14-33-20-23)35-31(38)21-36-15-12-26(13-16-36)34-30(37)18-22-5-2-1-3-6-22/h1-7,9-10,14,19-20,26,28-29H,8,11-13,15-18,21H2,(H,34,37)(H,35,38)
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n/an/a 36n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090397
PNG
(CHEMBL42620 | {1-[(6-Fluoro-1-pyridin-3-ylmethyl-1...)
Show SMILES CC(C)(C)OC(=O)NC1CCN(CC(=O)NC2CCc3cc(F)ccc3C2Cc2cccnc2)CC1
Show InChI InChI=1S/C28H37FN4O3/c1-28(2,3)36-27(35)31-22-10-13-33(14-11-22)18-26(34)32-25-9-6-20-16-21(29)7-8-23(20)24(25)15-19-5-4-12-30-17-19/h4-5,7-8,12,16-17,22,24-25H,6,9-11,13-15,18H2,1-3H3,(H,31,35)(H,32,34)
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n/an/a 37n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090391
PNG
(CHEMBL42437 | N-[4-(6-Fluoro-1-pyridin-3-ylmethyl-...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)[C@H]1CC[C@H](CNC(=O)c2ccccc2)CC1
Show InChI InChI=1S/C31H34FN3O2/c32-26-13-14-27-25(18-26)12-15-29(28(27)17-22-5-4-16-33-19-22)35-31(37)24-10-8-21(9-11-24)20-34-30(36)23-6-2-1-3-7-23/h1-7,13-14,16,18-19,21,24,28-29H,8-12,15,17,20H2,(H,34,36)(H,35,37)/t21-,24-,28?,29?
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n/an/a 39n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090404
PNG
(CHEMBL42020 | {1-[(6-Fluoro-1-pyridin-3-ylmethyl-1...)
Show SMILES CC(C)(C)OC(=O)NC1CCN(CC(=O)NC2CCc3cc(F)ccc3C2Cc2cccnc2)C1
Show InChI InChI=1S/C27H35FN4O3/c1-27(2,3)35-26(34)30-21-10-12-32(16-21)17-25(33)31-24-9-6-19-14-20(28)7-8-22(19)23(24)13-18-5-4-11-29-15-18/h4-5,7-8,11,14-15,21,23-24H,6,9-10,12-13,16-17H2,1-3H3,(H,30,34)(H,31,33)
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n/an/a 45n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090400
PNG
(CHEMBL46799 | {1-[(6-Fluoro-1-pyridin-3-ylmethyl-1...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CCC(CC1)NC(=O)Oc1ccccc1
Show InChI InChI=1S/C30H33FN4O3/c31-23-9-10-26-22(18-23)8-11-28(27(26)17-21-5-4-14-32-19-21)34-29(36)20-35-15-12-24(13-16-35)33-30(37)38-25-6-2-1-3-7-25/h1-7,9-10,14,18-19,24,27-28H,8,11-13,15-17,20H2,(H,33,37)(H,34,36)
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n/an/a 52n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090399
PNG
(CHEMBL42768 | N-(6-Methoxy-1-pyridin-3-ylmethyl-1,...)
Show SMILES COc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CCC(CC1)n1c2ccccc2[nH]c1=O
Show InChI InChI=1S/C31H35N5O3/c1-39-24-9-10-25-22(18-24)8-11-27(26(25)17-21-5-4-14-32-19-21)33-30(37)20-35-15-12-23(13-16-35)36-29-7-3-2-6-28(29)34-31(36)38/h2-7,9-10,14,18-19,23,26-27H,8,11-13,15-17,20H2,1H3,(H,33,37)(H,34,38)
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n/an/a 75n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090387
PNG
(4-(Phenylacetylamino-methyl)-cyclohexanecarboxylic...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)[C@H]1CC[C@H](CNC(=O)Cc2ccccc2)CC1
Show InChI InChI=1S/C32H36FN3O2/c33-27-13-14-28-26(19-27)12-15-30(29(28)17-24-7-4-16-34-20-24)36-32(38)25-10-8-23(9-11-25)21-35-31(37)18-22-5-2-1-3-6-22/h1-7,13-14,16,19-20,23,25,29-30H,8-12,15,17-18,21H2,(H,35,37)(H,36,38)/t23-,25-,29?,30?
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n/an/a 114n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090405
PNG
(2-[4-(3-tert-Butyl-ureido)-piperidin-1-yl]-N-(6-fl...)
Show SMILES CC(C)(C)NC(=O)NC1CCN(CC(=O)NC2CCc3cc(F)ccc3C2Cc2cccnc2)CC1
Show InChI InChI=1S/C28H38FN5O2/c1-28(2,3)33-27(36)31-22-10-13-34(14-11-22)18-26(35)32-25-9-6-20-16-21(29)7-8-23(20)24(25)15-19-5-4-12-30-17-19/h4-5,7-8,12,16-17,22,24-25H,6,9-11,13-15,18H2,1-3H3,(H,32,35)(H2,31,33,36)
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n/an/a 140n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090393
PNG
(4-[(3-Phenyl-ureido)-methyl]-cyclohexanecarboxylic...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)[C@H]1CC[C@H](CNC(=O)Nc2ccccc2)CC1
Show InChI InChI=1S/C31H35FN4O2/c32-25-13-14-27-24(18-25)12-15-29(28(27)17-22-5-4-16-33-19-22)36-30(37)23-10-8-21(9-11-23)20-34-31(38)35-26-6-2-1-3-7-26/h1-7,13-14,16,18-19,21,23,28-29H,8-12,15,17,20H2,(H,36,37)(H2,34,35,38)/t21-,23-,28?,29?
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n/an/a 170n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
Neuropeptide Y receptor type 5 ( NPY Y5)


(Homo sapiens (Human))
BDBM50090394
PNG
(CHEMBL44338 | N-(6-Fluoro-1-pyridin-3-ylmethyl-1,2...)
Show SMILES Fc1ccc2C(Cc3cccnc3)C(CCc2c1)NC(=O)CN1CCC(CC1)NC(=O)Nc1ccccc1
Show InChI InChI=1S/C30H34FN5O2/c31-23-9-10-26-22(18-23)8-11-28(27(26)17-21-5-4-14-32-19-21)35-29(37)20-36-15-12-25(13-16-36)34-30(38)33-24-6-2-1-3-7-24/h1-7,9-10,14,18-19,25,27-28H,8,11-13,15-17,20H2,(H,35,37)(H2,33,34,38)
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Article
PubMed
n/an/a 236n/an/an/an/an/an/a



The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell line


Bioorg Med Chem Lett 10: 1641-3 (2000)


Article DOI: 10.1016/s0960-894x(00)00311-5
BindingDB Entry DOI: 10.7270/Q2VQ31ZQ
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%