Compile Data Set for Download or QSAR
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Found 19 Enz. Inhib. hit(s) with all data for entry = 50010050
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090395(CHEMBL42762 | N-(6-Hydroxy-1-pyridin-3-ylmethyl-1,...)
Affinity DataIC50:  6nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090398(CHEMBL45199 | [4-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Affinity DataIC50:  16nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090403(CHEMBL43659 | {(S)-1-[(6-Fluoro-1-pyridin-3-ylmeth...)
Affinity DataIC50:  17nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090390(2-[4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperi...)
Affinity DataIC50:  22nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090402(CHEMBL296022 | N-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Affinity DataIC50:  25nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090388(CHEMBL42658 | N-{(S)-1-[(6-Fluoro-1-pyridin-3-ylme...)
Affinity DataIC50:  26nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090392(CHEMBL44886 | N-{1-[(6-Fluoro-1-pyridin-3-ylmethyl...)
Affinity DataIC50:  28nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090401(CHEMBL42031 | {(R)-1-[(6-Fluoro-1-pyridin-3-ylmeth...)
Affinity DataIC50:  30nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090396(CHEMBL44036 | [4-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Affinity DataIC50:  31nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090389(CHEMBL288763 | N-(6-Fluoro-1-pyridin-3-ylmethyl-1,...)
Affinity DataIC50:  36nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090397(CHEMBL42620 | {1-[(6-Fluoro-1-pyridin-3-ylmethyl-1...)
Affinity DataIC50:  37nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090391(CHEMBL42437 | N-[4-(6-Fluoro-1-pyridin-3-ylmethyl-...)
Affinity DataIC50:  39nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090404(CHEMBL42020 | {1-[(6-Fluoro-1-pyridin-3-ylmethyl-1...)
Affinity DataIC50:  45nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090400(CHEMBL46799 | {1-[(6-Fluoro-1-pyridin-3-ylmethyl-1...)
Affinity DataIC50:  52nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090399(CHEMBL42768 | N-(6-Methoxy-1-pyridin-3-ylmethyl-1,...)
Affinity DataIC50:  75nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090387(4-(Phenylacetylamino-methyl)-cyclohexanecarboxylic...)
Affinity DataIC50:  114nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090405(2-[4-(3-tert-Butyl-ureido)-piperidin-1-yl]-N-(6-fl...)
Affinity DataIC50:  140nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090393(4-[(3-Phenyl-ureido)-methyl]-cyclohexanecarboxylic...)
Affinity DataIC50:  170nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50090394(CHEMBL44338 | N-(6-Fluoro-1-pyridin-3-ylmethyl-1,2...)
Affinity DataIC50:  236nMAssay Description:Inhibition of binding of radioligand [125I]-PYY to the human Neuropeptide Y receptor type 5, using a stably transfected HEK293 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed