Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50036844
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50017702(1-(bis(4-fluorophenyl)methyl)-4-cinnamylpiperazine...)
Affinity DataIC50:  228nMAssay Description:Concentration required for 50% inhibitory effect on Dopamine receptor D2 determined in competition experiments with [3H]racloprideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50091592(7-{4-[Bis-(4-fluoro-phenyl)-methyl]-piperazin-1-yl...)
Affinity DataIC50:  1.69E+3nMAssay Description:Concentration required for 50% inhibitory effect on Dopamine receptor D2 determined in competition experiments with [3H]racloprideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50091591((2S)-1-(4-amino-2,3,5-trimethylphenoxy)-3-{4-[4-(4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required for 50% inhibitory effect on Dopamine receptor D2 determined in competition experiments with [3H]racloprideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed